PRIMAQUINE PHOSPHATE

PRIMAQUINE PHOSPHATE


Brand Names : Primachin phosphate; Primaquini diphosphas; Primaquinium phosphate; SN-13, 272.




It is an orange-red, odourless, crystalline, bitter powder, m.p. 197-198°. It is moderately soluble in water, insoluble in chloroform and ether. The aqueous solutions are acidic to litmus. The compound is protected from light.



Uses: Primaquine is antimalarial and effective against plasmodia parasite.

Adverse Effect


Primaquine is generally well tolerated at normal therapeutic doses. Adverse effects include abdominal cramps, gastric distress, nausea and vomiting, headache, visual disturbances, and pruritus.



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